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1
Synthese und Pharmakologie potenter 5-HT2A-Rezeptoragonisten mit N-2-Methoxybenzyl-Partialstruktur Entwicklung eines neuen Struktur-Wirkungskonzepts
Freien Universität Berlin
Ralf Heim
mmol
ht2a
ppm
abb
ch2cl2
och3
nmr
meoh
mhz
ausbeute
synthese
ch3
abs
rezeptoren
nh3
chinazolindion
feststoff
hcl
erfolgt
farblose
dmso
abschn
rezeptor
etoh
gelöst
cdcl3
experimenteller
freie
nh2
resp
mol
öl
derivate
chn
analog
gef
emax
aminoethyl
et2o
reduktive
affinität
hydrochlorid
pharmacol
synthetischer
zugabe
dimethoxyphenyl
pec50
benzyl
lösung
wirkung
Year:
2003
Language:
german
File:
PDF, 3.73 MB
Your tags:
0
/
4.0
german, 2003
2
Progress in Medicinal Chemistry 48
Academic Press, Elsevier
G. Lawton and D.R. Witty (Eds.)
receptor
ic50
motilin
ht6
binding
activity
compounds
inhibitors
appl
pct
bace
patent
abstr
assay
gastric
reported
antagonists
ligands
potent
clinical
drugs
rabbit
affinity
receptors
inhibition
ligand
potency
erythromycin
pec50
showed
studies
p110a
discovery
cellular
nh2
disclosed
patients
selectivity
molecule
mtor
target
agonists
μm
bioorg
pi3k
chemistry
analogues
derivatives
examples
peptide
Year:
2009
Language:
english
File:
PDF, 8.63 MB
Your tags:
0
/
0
english, 2009
3
Design, Synthesis and Pharmacological Evaluation of Certain GABA B Agonists: Dissertation
Mohamad Ibrahim Attia
ch3
phenyl
nmr
ester
reaction
receptors
ch2
ppm
amino
mixture
chloro
ethyl
methyl
gabab
harom
compounds
baclofen
synthesis
cdcl3
gaba
receptor
experimental
butenoic
solution
iodo
mmol
pentanoic
carom
hydrochloride
neat
binding
oc2h5
nh3
activity
aryl
ligand
tlc
discussion
ether
jab
evaporated
figure
theoretical
butanoic
pec50
stirred
gabaa
step
temperature
cooh
Year:
2003
Language:
english
File:
PDF, 2.27 MB
Your tags:
0
/
5.0
english, 2003
4
Infectivity and Drug Susceptibility Profiling of Different Leishmania-Host Cell Combinations
MDPI
Kyung-Hwa Baek
,
Laura Piel
,
Thibault Rosazza
,
Eric Prina
leishmania
infection
donovani
amazonensis
bmdm
amastigote
thp
figure
amastigotes
parasites
infected
susceptibility
promastigote
intracellular
hpi
vitro
infections
parasite
drugs
promastigotes
values
activity
assay
ec50
ssg
macrophages
observed
antileishmanial
phenotypic
miltefosine
showed
µm
compounds
leishmaniasis
pathogens
screening
assays
axenic
increase
species
discovery
macrophage
pvs
extracellular
supplementary
ampb
analysis
antimicrob
differentiated
j.h.n
Year:
2020
Language:
english
File:
PDF, 814 KB
Your tags:
0
/
0
english, 2020
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